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송규용,배기환,명창선,김문일,박용진,윤미영,김동희,Song Gyu Yong,Bae Ki Whan,Myung Chang-Seon,Jin Wen Yi,Park Yong Jin,Yun Mi Young,Kim Dong Hee 대한동의생리학회 2005 동의생리병리학회지 Vol.19 No.3
Antitumor and anti-metastatic effects of mineral powder(MP) were studied. In the present study, MP did not exhibit the any cytotoxic activity against leukemic cells such as L1210 and U937 tumor cell lines in vitro. Also, MP did not exhibit the any cytotoxic activity against solid cells such as A549 and B16-BL6 tumor cell lines in vitro. However, in vivo, MP exhibit a significant antitumor activity in BDF1 mice bearing Lewis lung carcinoma cells(LLC) with inhibition rates of 46 and $23\%$ at 200 and 100 mg/kg/day, respectively. Furthermore, in pulmonary colonization assay, MP exhibit the inhibitory effect of tumor metastasis. From these results, it was concluded that MP had antitumor and anti-metastatic activity suggesting its application for the prevention and treatment of cancer.
이지현,이재호,김현관,김의검,신귀남,조수현,명창선,김동희,윤미영,최용석,김성훈,송규용,Lee, Jee-Hyun,Lee, Jae-Ho,Kim, Hyun-Kwan,Kim, Eui-Geom,Shen, Gui-nan,Cho, Soo-Hyun,Myung, Chang-Seon,Kim, Dong-Hee,Yun, Mi-Young,Choi, Yong-Seok,Kim, Su 대한약학회 2006 약학회지 Vol.50 No.5
A novel series of 4-senecioyloxymethyl-6,7-dimethoxycoumarin, isolated from Crinum latifolium, was prepared by reacting 4-bromomethyl or 4-bromomethyl-6,7- dimethoxycoumarin with various carboxylic acids and examined for their anti-angiogenic activities in human umbilical vein endothelial cells (HUVECs). Among them, 4e, 4f, 4g and 4i with noncyclic moiety exhibited potent anti-angiogenic activity. However, compounds with cyclic moiety such as phenyl, pyridinyl, thiophenyl and furanyl group did not exhibit any anti-angiogenic activity. Also, compounds 4f and 4g which exhibited strong anti-angiogenic activity in a dose-dependent manner showed antitumor activity.
정상 식이 수컷 흰쥐에서 흑삼이 체중 및 지질에 미치는 영향
송규용(Gyu Yong Song),오한진(HAn Jin Oh),노성수(Seong Soo Roh),서영배(Young Bae Seo),박용진(Yong Jin Park),명창선(Chang-Seon Myung) 대한약학회 2006 약학회지 Vol.50 No.6
Previously, we have reported that black ginseng was produced by nine-time repeated steaming 5-year fresh ginsengs at 95℃ for 3 hr in pottery apparatus and drying at 60℃ for 12~36 hr and had an outstanding anticancer activity. This study was designed to examine the ability of black ginseng to suppress body weight gain and appetite, and to investigate the effect of black ginseng on lipid profile in male rats fed normal diets. The extract of black ginseng was administered daily for 3 weeks, and the changes of body weight and food intake were measured. After administering the extracts for 3 weeks, the fat weight and serum lipid levels were also measured. Black ginseng persistently suppressed weigh gain and food intake was also reduced, but not significantly. The weight of both epididymal and abdominal fats was decreased in black ginseng-treated rats. Serum triglyceride level in rats administered with black ginseng was also significantly lowered. Therefore, these results reveal that the repeated administration of black ginseng causes a suppression body weigh gain by decreasing triglyceride level in blood and body fat deposit.