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Lipoxygenase Inhibitory Constituents from Indigofera oblongifolia
Ahsan Sharif,Ejaz Ahmed,Abdul Malik,Naheed Riaz,Nighat Afza,Sarfraz Ahmad Nawaz,Muhammad Arshad,Muhammad Raza Shah,Muhammad Iqbal Choudhary 대한약학회 2005 Archives of Pharmacal Research Vol.28 No.7
Indigin, alkylated xanthene (1) and indigoferic acid (2) have been isolated from the chloroform soluble fraction of Indigofera oblongifolia, along with β-sitosterol (3) and 3-hydroxybenzoic acid (4), which are reported for the first time from this species. Their structures were determined through spectroscopic techniques. Both the new compounds 1 and 2 showed significant activity against enzyme lipoxygenase, while 2 further showed moderate inhibition against BChE.
Muhammad Ahsan Sami,Muhammad Umar Masood,Muhammad Waqar,Muhammad Mujtaba,Abrahim Ali Shah,Nasir Rashid,Mohsin I. Tiwana,Javaid Iqbal,Adnan Shujah 제어로봇시스템학회 2017 제어로봇시스템학회 국제학술대회 논문집 Vol.2017 No.10
This paper presents an application of a novel approach for detecting and tracking an object with a 2 DOF robotic manipulator which can be equipped with an array of electrically controlled actuators. The said approach utilizes the Image Based Visual Servoing (IBVS) technique. The developed system is able to determine the object pose in real time from features in the image. Object is detected using shaped based approach algorithms of image processing. The position and orientation of the world coordinates of the object being tracked are calculated from the coordinates of the object in image plane using camera’s intrinsic and extrinsic parameters. Experimental results demonstrate the effectiveness of this proposed approach.
Lipoxygenase Inhibitory Constituents from Indigofera oblongifolia
Sharif, Ahsan,Ahmed, Ejaz,Malik, Abdul,Riaz, Naheed,Afza, Nighat,Nawaz, Sarfraz Ahmad,Arshad, Muhammad,Shah, Muhammad Raza,Chaudhary, Muhammad Iqbal The Pharmaceutical Society of Korea 2005 Archives of Pharmacal Research Vol.28 No.7
Indigin, alkylated xanthene (1) and indigoferic acid (2) have been isolated from the chloroform soluble fraction of Indigofera oblongifolia, along with $\beta$-sitosterol (3) and 3-hydroxybenzoic acid (4), which are reported for the first time from this species. Their structures were determined through spectroscopic techniques. Both the new compounds 1 and 2 showed significant activity against enzyme lipoxygenase, while 2 further showed moderate inhibition against BChE.
Channel Allocation in Multi-radio Multi-channel Wireless Mesh Networks: A Categorized Survey
( Saleem Iqbal ),( Abdul Hanan Abdullah ),( Khalid Hussain ),( Faraz Ahsan ) 한국인터넷정보학회 2015 KSII Transactions on Internet and Information Syst Vol.9 No.5
Wireless mesh networks are a special type of broadcast networks which cover the qualifications of both ad-hoc as well as infrastructure mode networks. These networks offer connectivity to the last mile through hop to hop communication and by comparatively reducing the cost of infrastructure in terms of wire and hardware. Channel assignment has always been the focused area for such networks specifically when using non-overlapping channels and sharing radio frequency spectrum while using multiple radios. It has always been a challenge for mesh network on impartial utilization of the resources (channels), with the increase in users. The rational utilization of multiple channels and multiple radios, not only increases the overall throughput, capacity and scalability, but also creates significant complexities for channel assignment methods. For a better understanding of research challenges, this paper discusses heuristic methods, measurements and channel utilization applications and also examines various researches that yield to overcome this problem. Finally, we highlight prospective directions of research.
Design and Development of a Semi-Autonomous Stair Climbing Robotic Platform For Rough Terrains
Muhammad Umar Masood,Muhammad Ahsan Sami,Haris Sohail,Muhammad Mujtaba,Muhammad Abubakar Siddique,Hashir Akram,Nasir Rashid,Mohsin I. Tiwana,Javaid Iqbal 제어로봇시스템학회 2017 제어로봇시스템학회 국제학술대회 논문집 Vol.2017 No.10
This paper presents the design of a stair climbing fixed flipper unmanned ground vehicle (UGV) for urban search and rescue purposes. Mobile flippers are being used in certain UGVs for enhanced mobility in rough terrains, however, the control algorithm of these platforms is complex. To add this enhanced mobility in the UGV and to reduce the intricacy of the control algorithm, anterior end of the tracks are lifted up which enables the UGV to pass over obstacles with relative ease. To prevent the rollover of UGV while moving on an inclined surface, an image processing algorithm was developed which halts the motion of UGV if the calculated slope exceeds the threshold value with a maximum error of about 8%. Furthermore, left and right track velocities along with the turn radius were also calculated.
Characterization and Comparative Evaluation of Milk Protein Variants from Pakistani Dairy Breeds
Iqra Yasmin,Rabia Iqbal,Atif Liaqat,Wahab Ali Khan,Muhamad Nadeem,Aamir Iqbal,Muhammad Farhan Jahangir Chughtai,Syed Junaid Ur Rehman,Saima Tehseen,Tariq Mehmood,Samreen Ahsan,Saira Tanweer,Saima Naz 한국축산식품학회 2020 한국축산식품학회지 Vol.40 No.5
The aim of study was to scrutinize the physicochemical and protein profile of milk obtained from local Pakistani breeds of milch animals such as Nilli-Ravi buffalo, Sahiwal cow, Kajli sheep, Beetal goat and Brela camel. Physicochemical analysis unveiled maximum number of total solids and protein found in sheep and minimum in camel. Buffalo milk contains the highest level of fat (7.45%) while camel milk contains minimum (1.94%). Ash was found maximum in buffalo (0.81%) and sheep (0.80%) while minimum in cow’s milk (0.71%). Casein and whey proteins were separated by subjecting milk to isoelectric pH and then analyzed through sodium dodecyl sulphate-polyacrylamide gel electrophoresis (SDS-PAGE). The results showed heterogeneity among these species. Different fractions including αS1, αS2, κ-casein, β-casein and β-lactoglobulen (β-Lg) were identified and quantitatively compared in all milk samples. Additionally, this electrophoretic method after examining the number and strength of different protein bands (αS1, αS2, β- CN, α-LAC, BSA, and β-Lg, etc.), was helpful to understand the properties of milk for different processing purposes and could be successfully applied in dairy industry. Results revealed that camel milk was best suitable for producing allergen free milk protein products. Furthermore, based on the variability of milk proteins, it is suggested to clarify the phylogenetic relationships between different cattle breeds and to gather the necessary data to preserve the genetic fund and biodiversity of the local breeds. Thus, the study of milk protein from different breed and species has a wide range of scope in producing diverse protein based dairy products like cheese.
Synchronous Reference Frame Theory Based Intelligent Controller for Current THD Reduction
Al-Ammar Essam A.,Ul Haq Azhar,Iqbal Ahsan,Ko Wonsuk,Jalal Marium,Anjum Muhammad Almas,Choi Hyeong-Jin,Kang Hyun-Koo 대한전기학회 2021 Journal of Electrical Engineering & Technology Vol.16 No.6
Concerns related to current harmonics have gained increased attention in recent years due to technological advancement in power electronics and the proliferation of non-linear loads in power distribution system. It has become challenging to limit current total harmonic distortion (THD) at consumer end mainly due to increased penetration of intermittent switching based non-linear loads. Shunt active power fi lter (SAPF) is considered a marvelous power electronics device to tackle consumer side current harmonics. This paper presents a synchronous reference frame (SRF) based improved control method for compliant working of SAPF to reduce current harmonics in the distribution network with same and diff erent THD levels in three phases. This research work investigates an eff ectual DC link voltage control technique linked with SRF based control of SAPF to eff ectively mitigate current harmonics. A fuzzy logic-based automatic switch (FLBAS) is designed according to the THD standards of IET and IEEE for real-time controlling of SRF based control of SAPF. In addition, S-plane stability analysis of the proposed control scheme is performed using the model of SAPF’s inverter. It is established that the closed-loop system is asymptotically stable with the proposed control scheme. The presented simulation results validate the eff ectiveness of the proposed control technique for SAPF robustly.
Raza, Rabia,Saeed, Aamer,Arif, Mubeen,Mahmood, Shamsul,Muddassar, Muhammad,Raza, Ahsan,Iqbal, Jamshed Blackwell Publishing Ltd 2012 Chemical biology & drug design Vol.80 No.4
<P>On the basis of the observed biological activity of the coumarins, a new set of 3‐thiazolocoumarinyl Schiff‐base derivatives with chlorine, hydroxy and methoxy functional group substitutions were designed and synthesized. These compounds were tested against acetylcholinesterase from <I>Electrophorus electricus</I> and butyrylcholinesterase from horse serum and their structure–activity relationship was established. Studies revealed them as the potential inhibitors of cholinesterase (acetylcholinesterase and butyrylcholinesterase). The <B>3f</B> was found to be most potent against acetylcholinesterase with <I>K</I><SUB>i</SUB> value of 1.05 ± 0.3 μ<SMALL>m</SMALL> and <B>3l</B> showed excellent inhibitory action against butyrylcholinesterase with <I>K</I><SUB>i</SUB> value of 0.041 ± 0.002 μ<SMALL>m</SMALL>. The synthesized compounds were also docked into the active sites of the homology models of acetylcholinesterase and butyrylcholinesterase to predict the binding modes of these compounds. It was predicted that most of the compounds have similar binding modes with reasonable binding affinities. Our docking studies have also shown that these synthesized compounds have better interaction patterns with butyrylcholinesterase over acetylcholinesterase. The main objective of the study was to develop new potent and selective compounds, which might be further optimized to prevent the progression of the Alzheimer’s disease and could provide symptomatic treatment.</P>