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Inhibitory Activity of Plantago major L. on Angiotensin I-converting Enzyme
Nguyen Xuan Nhiem,김영호,Bui Huu Tai,Phan Van Kiem,Chau Van Minh,Nguyen Xuan Cuong,Nguyen Huu Tung,Vu Kim Thu,Trinh Nam Trung,Hoang Le Tuan Anh,조성훈,장해동,권영인 대한약학회 2011 Archives of Pharmacal Research Vol.34 No.3
Eight compounds were isolated from methanol extract of Plantago major L. leaves and investigated for their ability to inhibit angiotensin I-converting enzyme activity. Among them, compound 1 showed the most potent inhibition with rate of 28.06 ± 0.21% at a concentration of 100 μM. Compounds 2 and 8 exhibited weak activities. These results suggest that compound 1 might contribute to the ability of P. major to inhibit the activity of angiotensin I- converting enzyme.
Chemical Constituents of the Morinda tomentosa Leaves and their α-Glucosidase Inhibitory Activity
Vu, Huong Giang,Ninh, Khac Ban,Nguyen, Xuan Nhiem,Phan, Van Kiem,Chau Van, Minh,Hoang, Le Tuan Anh,Pham, Hai Yen,Bui, Huu Tai,Nguyen, Xuan Cuong,Nguyen, Hoai Nam,Kim, Seung Hyun,Kwon, Young-In,Kim, Yo Korean Chemical Society 2013 Bulletin of the Korean Chemical Society Vol.34 No.5
Tobacco Control Policies in Vietnam: Review on MPOWER Implementation Progress and Challenges
Hoang, Van Minh,Tran, Thu Ngan,Vu, Quynh Mai,Nguyen, Thi Tuyet My,Le, Hong Chung,Vu, Duy Kien,Tran, Tuan Anh,Nguyen, Bao Ngoc,Vu, Van Giap,Nguyen, Manh Cuong,Pham, Duc Manh,Kim, Bao Giang Asian Pacific Journal of Cancer Prevention 2016 Asian Pacific journal of cancer prevention Vol.17 No.no.sup1
In Vietnam, the WHO Framework Convention on Tobacco Control (WHO FCTC) took effect in March 2005 while MPOWER has been implemented since 2008. This paper describes the progress and challenges of implementation of the MPOWER package in Vietnam. We can report that, in term of monitoring, Vietnam is very active in the Global Tobacco Surveillance System, completing two rounds of the Global Adult Tobacco Survey (GATS) and three rounds of the Global Youth Tobacco Survey (GYTS). To protect people from tobacco smoke, Vietnam has issued and enforced a law requiring comprehensive smoking bans at workplaces and public places since 2013. Tobacco advertising and promotion are also prohibited with the exception of points of sale displays of tobacco products. Violations come in the form of promotion girls, corporate social responsibility activities from tobacco manufacturers and packages displayed by retail vendors. Vietnam is one of the 77 countries that require pictorial health warnings to be printed on cigarette packages to warn about the danger of tobacco and the warnings have been implemented effectively. Cigarette tax is 70% of factory price which is equal to less than 45% of retail price and much lower than the recommendation of WHO. However, Vietnam is one of the very few countries that require manufacturers and importers to make "compulsory contributions" at 1-2% of the factory price of cigarettes sold in Vietnam for the establishment of a Tobacco Control Fund (TCF). The TCF is being operated well. In 2015, 67 units of 63 provinces/cities, 22 ministries and political-social organizations and 6 hospitals received funding from TCF to implement a wide range of tobacco control activities. Cessation services have been starting with a a toll-free quit-line but need to be further strengthened. In conclusion, Vietnam has constantly put efforts into the tobacco control field with high commitment from the government, scientists and activists. Though several remarkable achievements have been gained, many challenges remain. To overcome those challenges, implementation strategies that take into account the contextual factors and social determinants of tobacco use in Vietnam are needed.
Triterpenoids from aerial parts of Glochidion eriocarpum.
Thu, Vu Kim,Kiem, Phan Van,Yen, Pham Hai,Nhiem, Nguyen Xuan,Tung, Nguyen Huu,Cuong, Nguyen Xuan,Minh, Chau Van,Huong, Hoang Thanh,Lau, Trinh Van,Thuan, Ngo Thi,Kim, Young Ho Natural Product Communications 2010 Natural product communications Vol.5 No.3
<P>From the aerial parts of Glochidion eriocarpum, a new triterpene, glochieriol (1), three new triterpenoid saponins, glochieriosides C - E (2 - 4), together with four known triterpenes (glochidonol, glochidiol, lupeol, and 3-epi-lupeol) were isolated by using combined chromatographic separations. The structures of the new compounds were elucidated on the basis of spectroscopic data, including FTICR-MS, 1D and 2D NMR.</P>
Vu Thi Yen,Wang Yao Nan,Pham Van Cuong,Nguyen Xuan Quynh,Vu Huu Thich 제어·로봇·시스템학회 2017 International Journal of Control, Automation, and Vol.15 No.6
In this paper, a robust adaptive control method based on Dynamic Structure Fuzzy Wavelet Neural Networks(FWNNs) system is presented for trajectory tracking control of industrial robot manipulators (IRM) withuncertainties and disturbances via adaptive sliding mode control (SMC). Four layer FWNNs in the Dynamic structureFWNNs is constructed on the basis of fuzzy rules which associates with wavelet function in the consequentpart, to compensate for structured and unstructured uncertainties and model complex processes. However, it isdifficult to design a suitable control scheme to achieve the required approximation errors, such as friction forces,external disturbances error and parameter variations. To deal with the mentioned problems, all the parameters of theDynamic structure FWNNs system are tuned on-line by an adaptive learning algorithm, and adaptive robust controllaws are determined by Lyapunov stability theorem. By using Dynamic structure FWNNs, this control systemcould achieve desired tracking performance, the stability and robustness of the closed-loop manipulators system areguaranteed. In addition, the simulations and experimental performed on a three-link IRM are provided in comparisonwith wavelet network control (WNC) and adaptive Fuzzy control (AFC) to demonstrate the effectiveness androbustness of the proposed Dynamic structure FWNNs methodology.
Cytotoxic Oleane-type Triterpene Saponins from Glochidion eriocarpum
Nguyen Xuan Nhiem,김영호,Vu Kim Thu,Phan Van Kiem,Chau Van Minh,Bui Huu Tai,TRANHONG QUANG,Nguyen Xuan Cuong,Pham Hai Yen,Hye-Jin Boo,강정일,강희경 대한약학회 2012 Archives of Pharmacal Research Vol.35 No.1
The anticancer activity of ten compounds from the aerial parts of Glochidion eriocarpum were evaluated on two human cancer cell lines, HL-60 and HCT-116. Compounds 1-4 displayed highly potent cytotoxic activity on the HCT-116 cancer cell line with IC50 values ranging of 0.41~1.16 μM. Compounds 1-4 significantly inhibited the HL-60 cell line with IC50 values ranging of 4.51~6.33 μM. These results suggested that the benzoyl group at the C-22 position in oleane-type triterpene saponins was essential for cytotoxicity towards tumor cells. Moreover, compounds 2 and 3 showed more potent cytotoxicity than compounds 1 and 4 against HL-60 and HCT-116 cells. With respect to the mechanism underlying cytotoxicity, compounds 1-4 increased chromatin condensation, a typical apoptotic characteristic in HL-60 and HCT-116 cells. In the mechanism of apoptosis induction, compounds 1-4 reduced Bcl-2expression, whereas the expression of Bax was increased compared to controls in HCT-116 cells. In addition, compounds 1-4 decreased the level of procaspase-3. The cleavage of poly (ADP-ribose) poly merase (PARP), a vital substrate of effector caspase, was observed in HCT-116 cells. Furthermore, the induction of apoptosis was also accompanied by an activation of extracellular signal-regulated kinase (ERK) and p38 kinase in HCT-116 cells. These findings provide evidence demonstrating that the pro-apoptotic effects of compounds 1-4 are mediated through the activation of ERK and p38 in HCT-116 cells.
Hoang, Van Minh,Le, Hong Chung,Kim, Bao Giang,Duong, Minh Duc,Nguyen, Duc Hinh,Vu, Quynh Mai,Nguyen, Manh Cuong,Pham, Duc Manh,Ha, Anh Duc,Yang, Jui-Chen Asian Pacific Journal of Cancer Prevention 2016 Asian Pacific journal of cancer prevention Vol.17 No.no.sup1
Two years after implementation of the graphic health warning intervention in Vietnam, it is very important to evaluate the intervention's potential impact. The objective of this paper was to predict effects of graphic health warnings on cigarette packages, particularly in reducing cigarette demand and smoking-associated deaths in Vietnam. In this study, a discrete choice experiment (DCE) method was used to evaluate the potential impact of graphic tobacco health warnings on smoking demand. To predict the impact of GHWs on reducing premature deaths associated with smoking, we constructed different static models. We adapted the method developed by University of Toronto, Canada and found that GHWs had statistically significant impact on reducing cigarette demand (up to 10.1% through images of lung damage), resulting in an overall decrease of smoking prevalence in Vietnam. We also found that between 428,417- 646,098 premature deaths would be prevented as a result of the GHW intervention. The potential impact of the GHW labels on reducing premature smoking-associated deaths in Vietnam were shown to be stronger among lower socio-economic groups.
Nhiem, Nguyen Xuan,Kiem, Phan Van,Minh, Chau Van,Tai, Bui Huu,Cuong, Nguyen Xuan,Thu, Vu Kim,Anh, Hoang Le Tuan,Jo, Sung-Hoon,Jang, Hae-Dong,Kwon, Young-In,Kim, Young Ho The Pharmaceutical Society of Japan 2010 Chemical & pharmaceutical bulletin Vol.58 No.10
<P>One new monoterpenoid glycoside, myresculoside (<B>1</B>), and eleven known compounds, were isolated from methanol extract of <I>Myrica esculenta</I> leaves by repeated column chromatography. The effects of these compounds on angiotensin I-converting enzyme (ACE) inhibition were investigated. Compounds <B>3</B> and <B>4</B> showed the most potent ACE inhibition with rates of 29.97% and 25.63% at concentration of 100 μ<SMALL>M</SMALL>, respectively. Compounds <B>5</B>, <B>6</B>, and <B>11</B> showed weak activity with inhibitory rates of 0.07—1.41% at concentration of 100 μ<SMALL>M</SMALL>.</P>