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천연물로부터의 세포내 효소 활성 조절물질의 탐색 및 기능 연구: 갈근의 알코을 탈수소효소 저해 활성 성분
이현주(Hyun Joo Lee),오민아(Min Ah Oh),최영희(Young Hui Choi),이강만(Kang Min Lee) 대한약학회 2001 약학회지 Vol.45 No.5
Puerariae Radix is one of the medicinal plants used in oriental medicine for hangover. It has been claimed for several pharmacological effects including anti-alcohol abuse, antidipsotropic activity and anti-alcohol intoxication. In connection with Puerariae Radix effects, an activity-guided purification of active substance on alcohol dehydrogenase (ADH) was carried-out. The most active compound was isolated as puerarin (C21H2OO9), molecular weight 416. Puerarin inhibited ADH noncompetitively against ethanol or NAD+.
이현주,오민아,최영희,이강만 梨花女子大學校 藥學硏究所 2001 藥學硏究論文集 Vol.- No.10
Puerariae Radix is one of the medicinal plants used in oriental medicine for hangover. It has been claimed for several pharmacological effects including anti-alchol abuse, antidipsotropic activity and anti-alcohol intoxication. In connection with Puerariae Radix effects, an activity-guided purification of active substance on alcohol dehydrogenase(ADH) was carried-out. The most active compound was isolated as puerarin (C_21H_20O_9), molecular weight 416. Puerarin inhibited ADH noncompetitively against ethanol or NAD^+