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Qing-Qing Dong,Qiu-Tong Wang,Lei Wang,Ya-Xin Jiang,Mei-Ling Liu,Hai-Jie Hu,Yong Liu,Hao Zhou,Hong-Peng He,Tong-Cun Zhang,Xuegang Luo 한국식품과학회 2018 Food Science and Biotechnology Vol.27 No.4
Sulforaphane (SFN), a natural compound derived from cruciferous vegetables, has been proved to possess potent anti-cancer activity. SMYD3 is a histone methyltransferase which is closely related to the proliferation and migration of cancer cells. This study showed that SFN could dose-dependently induce cell cycle arrest, stimulate apoptosis, and inhibit proliferation and migration of gastric carcinoma cells. Accompanied with these anticancer effects, SMYD3 and its downstream genes, myosin regulatory light chain 9, and cysteine-rich angiogenic inducer 61, was downregulated by SFN. Furthermore, overexpression of SMYD3 via transfection could abolish the effects of SFN, suggesting that SMYD3 might be an important mediator of SFN. To the best of our knowledge, this is the first report describing the role of SMYD3 in the anti-cancer of SFN. These findings might throw light on the development of novel anti-cancer drugs and functional food using SFN-rich cruciferous vegetables.
Optimization of preparation and properties of Gardenia yellow pigment-loaded alginate beads
Yong Liu,Qing Zhou,Yan-Mei He,Xiu-Yun Ma,Lin-Na Liu,Yong-Jian Ke 한국화학공학회 2021 Korean Journal of Chemical Engineering Vol.38 No.8
Gardenia yellow pigment (GYP) loaded alginate beads were prepared by the ionic gelation technique, and the preparation parameters were optimized by response surface methodology for high encapsulation efficiency. The optimized parameters were alginate concentration of 3.3%, CaCl2 concentration of 2.4%, and GYP concentration of 3.2mg/mL, under which the encapsulation efficiency was 73.61%. The surface morphology and bead size analysis showed that the GYP-loaded alginate beads had a roughly spherical morphology with a wrinkled surface, and their average diameter was 0.87 mm. In vitro release test revealed that the GYP release had a pH-dependent release profile and a two-step release process. The Rigter-Peppas model was the most proper model to assess the GYP release from alginate beads. The release mechanism of GYP at pH 1.2 and 7.4 was non-Fickian transport and case-II transport, respectively. The 2,2-diphenyl-1-picrylhydrazyl assay indicated that the encapsulated GYP had effectively maintained 82.56% of the antioxidant activity.
Effects of Ozone on the Cytomembrane and Ultrastructure of Pseudomonas aeruginosa
Yong-qing Zhang,Qing-ping Wu,Ju-mei Zhang,Xiu-hua Yang 한국식품과학회 2015 Food Science and Biotechnology Vol.24 No.3
The ozone impact on Pseudomonas aeruginosa ATCC27853 cells was studied. Ozone-induced loss of K+, Mg2+, and ATP was measured using inductively coupled plasma/mass spectrometry and a bioluminescence assay. Maximum releases of K+ and Mg2+ were achieved at 0.37 mg/L of ozone after 2 min with a killing rate of culturable bacteria greater than 93%. Maximum release of ATP was attained at 0.42 mg/L of ozone after 3 min. Transmission electron microscopy showed that shapes of treated cells were integrated, but cytoplasmic agglutinations and vacuoles appeared. Ozone treatment caused lysis of P. aeruginosa cells to be sensitive to sodium dodecyl sulfate, insensitive to NaOH, and subject to inactivation by proteinase K. A combined action of cytoplasm agglutination, protein denaturation, and membrane permeabilization, rather than cell lysis, leads to non-culturability of P. aeruginosa cells.
Synthesis, Antibacterial Activity, and Structure–Activity Relationship of Fusaric Acid Analogs
Qing-Yan Zhang,Yang Fei‐Yu,Liao Shang‐Gao,Wang Bing,Li Rui,Dong Yong‐Xi,Zhou Meng,Yang Yuan‐Yong,Xu Guo‐Bo 대한화학회 2021 Bulletin of the Korean Chemical Society Vol.42 No.4
Forty-one fusaric acid analogs possessing a pyridine carboxylic acid scaffold have been synthesized. The antibacterial activity results demonstrated that compounds 5b, 7b, 8c, and 8d displayed strong antibacterial activities against Staphylococcus aureus ATCC25923 with minimum inhibitory concentrations (MICs) of 4–16 μg/mL. Molecular docking study indicated that these compounds have strong hydrogen-bonding interactions with TyrRS. Meanwhile, 8c and 8d showed promising antibacterial activities against Pseudomonas aeruginosa ATCC9027. Compound 4 exhibited pronounced antibacterial activities against a clinically isolated multidrug-resistant strain of Escherichia coli (MIC: 64 μg/mL as compared 64 μg/mL of levofloxacin and 1024 μg/mL of ceftriaxone sodium). Moreover, compound 17e displayed strong synergistic antibacterial effect with levofloxacin against the multidrug-resistant strain, decreasing the MIC value of levofloxacin to 1/16 of its original MIC. No obvious cytotoxic activities against LO2 was observed for compounds 4, 5b, 8c, 8d, 17d, and 17e at 50 μM. The preliminary structure–activity relationship of fusaric acid analogs was also discussed.
Qing-Yong Wang,He-Rui Zhang,Yu Gao,Rong-Hai Li,Xiao-Hong Shang 대한진단검사의학회 2017 Annals of Laboratory Medicine Vol.37 No.5
Dear Editor, Persistent infection with human papillomavirus (HPV) is the main cause of cervical cancer. Screening of cervical specimens for high-risk human papillomaviruses (HR-HPV) has become a routine part of patient care in most countries. The Roche cobas 4800 system (Roche Molecular Systems Inc., Pleasanton, CA, USA), a fully automated system that uses in vitro qualitative real-time PCR technology, displays high sensitivity and specificity for HR-HPV detection [1]. However, a small proportion of invalid results may occur in specimens showing mucopurulent discharge because of pipetting errors, clot formation, or failed amplification, which could cause a delay in the results and lead to additional waiting time for patients and extra work hours for staff, although most cases are resolved by vortexing the specimens and retesting. To the best of our knowledge, no researcher has tried to overcome this problem by pretreating specimens with an appropriate concentration of Sputasol (Oxoid Ltd., Basingstoke, United Kingdom); Sputasol (dithiothreitol 1.4%) has been used to aid culturing and DNA extraction from sputum specimens in some laboratories [2]. Here, we propose a standard method to improve HR-HPV detection without affecting the performance of the cobas 4800 HPV system.
Regional Differences and Variability on Enterprise Management Performance: A case in China
Yong qing Xiong,Yun wen Feng,Xiao hong Chen 사람과세계경영학회 2013 Global Business and Finance Review Vol.18 No.2
This paper measures variation in the economic performance of firms using the entropy weight method and cluster analysis. Regional differences and changes in the trend of listed companies' management performance are analyzed in China's four economic regions and 31 provinces from 2006 to 2010, the Eleventh Five Year period. We show that the listed companies' management performance in four economic regions presents a ladder type distribution with large swings and different trends over time. Moreover, there is a large difference in listed companies' management performance across provinces and some provinces have abnormal fluctuations. It is indicated that differences in industrial structures across regions are the main factor determining regional differences in economic development and the variability of enterprise management performance. So from the perspective of policy and institution, some suggestions are advanced to promote integrated development of all regions. In addition, the research results can provide governments at all levels with systematic reference information to formulate a coordinated, sustainable development policy for different regional economies.
Adaptive Fuzzy Control with Compressors and Limiters for a Class of Uncertain Nonlinear Systems
Yong-Qing Fan,Yin-He Wang,Yun Zhang,Qin-Ruo Wang 제어·로봇·시스템학회 2013 International Journal of Control, Automation, and Vol.11 No.3
This paper proposes a novel adaptive fuzzy control design for a class of nonlinear uncertain systems. The definition of compressor and limiter with adjustable parameters is introduced at beginning, and then updated laws of parameters of the compressor and estimate values of fuzzy approximation accuracies are utilized to synthesize stable adaptive controllers. The most advantage of designing adaptive fuzzy controller is neglectful of the logic structure of fuzzy logic systems, which make de-signer focus on parameters of the compressor, limiter and fuzzy approximation accuracies. This adap-tive fuzzy control method can not only reduce the number of on-line updated parameters but also guarantee states of the closed-loop system to be uniformly ultimately bounded (UUB). Simulation results demonstrate the effectiveness of the control scheme in this paper.
The Research on Chinese Enterprises` "Going Out" Model with Headquarters Economy
ZHANG Yong-qing,Jl xiu-jun 한국도시행정학회 2013 한국도시행정학회 학술발표대회 논문집 Vol.2013 No.9
Because of the effect of industrial division and economic globalization being increasingly apparent, industry chain become globalization tendency. On the basis of the research on global value chain, we summarize the development and advantage of headquarters economy. And then we find out the smiling curve relation of headquarters economy and global value chain. So we come up with three phases. In the end, we put forward Chinese enterprises" "going out" models which are functions headquarters abroad and manufacture base abroad.