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( Lin Ye ),( Yang Xin ),( Zhi-yuan Wu ),( Hai-jian Sun ),( De-jian Huang ),( Zhi-qin Sun ) 한국미생물 · 생명공학회 2022 Journal of microbiology and biotechnology Vol.32 No.1
Luteolin is a common dietary flavone possessing potent anti-inflammatory activities. However, when administrated in vivo, luteolin becomes methylated by catechol-O-methyltransferases (COMT) owing to the catechol ring in the chemical structure, which largely diminishes its anti-inflammatory effect. In this study, we made a modification on luteolin, named LUA, which was generated by the chemical reaction between luteolin and 2,2'-azobis(2-amidinopropane) dihydrochloride (AAPH). Without a catechol ring in the chemical structure, this new flavone could escape from the COMT-catalyzed methylation, thus affording the potential to exert its functions in the original form when administrated in the organism. Moreover, an LPS-stimulated RAW cell model was applied to detect the anti-inflammatory properties. LUA showed much more superior inhibitory effect on LPS-induced production of NO than diosmetin (a major methylated form of luteolin) and significantly suppressed upregulation of iNOS and COX-2 in macrophages. LUA treatment dramatically reduced LPS-stimulated reactive oxygen species (ROS) and mRNA levels of pro-inflammatory mediators such as IL-1β, IL-6, IL-8 and IFN-β. Furthermore, LUA significantly reduced the phosphorylation of JNK and p38 without affecting that of ERK. LUA also inhibited the activation of NF-κB through suppression of p65 phosphorylation and nuclear translocation.
Liposome Formulation of Paclitaxel with Enhanced Solubility and Stability
Yang, Tao,Cui, Fu-De,Choi, Min-Koo,Lin, Hongxia,Chung, Suk-Jae,Shim, Chang-Koo,Kim, Dae-Duk Informa Healthcare 2007 DRUG DELIVERY Vol.14 No.5
<P> Despite its strong antitumor activity, paclitaxel (Taxol®) has limited clinical applications due to its low aqueous solubility and hypersensitivity caused by Cremophor® EL and ethanol which is the vehicle used in the current commercial product. In an attempt to develop a pharmaceutically acceptable formulation that could replace Taxol®, a paclitaxel incorporated liposome has been constructed to improve solubility and physicochemical stability. The effect of various components of the liposome, including cholesterol and lipid, on the solubility and entrapment efficiency (EE) of paclitaxel was systematically investigated. The results showed that 5% (v/v) of polyethylene glycol 400 in the hydration medium of liposome significantly increased the solubility (up to 3.39 mg/mL) as well as the EE and the paclitaxel content in the liposome formulation composed of 10% (w/v) of S100PC with cholesterol (cholesterol-to-lipid molar ratio = 10:90). When sucrose (sugar-to-lipid molar ratio = 2.3) was added as a lyoprotectant during the freeze-drying of the liposome, physicochemical stability of liposome was significantly improved. Moreover, the cytotoxicity of the final liposome formulation against MDA-MB-231 human breast cancer cell line was not significantly different from that of Taxol®. The enhanced aqueous solubility as well as the physicochemical stability of paclitaxel in the liposome formulation developed in this study could be a safer and effective alternative to the Cremophor® EL and ethanol formulation.</P>
De Sun,Ping Yang,Lin Li,Hai-Hua Yang,Bing-Bing Li 한국화학공학회 2014 Korean Journal of Chemical Engineering Vol.31 No.10
A novel PDMS-PTFE/PVDF hollow fiber composite membrane using PTFE-PDMS as the top active layerand PVDF hollow fiber as the support layer was prepared for the pervaporation of chloroform from water. Sorptionand diffusion behaviors of chloroform and water in PDMS-PTFE membranes, which had different PTFE content, wereinvestigated. The results showed that with increasing PTFE content from 0 wt% to 40 wt%, chloroform/water idealseparation factor first increased and then decreased, and permeabilities of both chloroform and water increased. Forthe 30% PTFE-PDMS membrane, when feed temperature ranged from 40 oC to 60 oC, permeabilities of both chloroformand water increased, but ideal separation factor for chloroform/water first increased and then decreased. Effects of op-erating conditions, such as feed flow rate, active layer thickness, feed concentration and feed temperature, on PV per-formances of the 30% PDMS-PTFE/PVDF hollow fiber membrane for the pervaporation of chloroform-water mixtureswere studied. Examination showed that concentration polarization on the membrane surface occurred when feed flowrate was less than 3,000 mL/min. With the increase in active layer thickness from 13.8 to 78.0 µm, chloroform fluxand water flux dropped from 21 to 13 g·h−1·m−2and from 93 to 22 g·h−1·m−2, respectively, but the separation factorincreased from 1494 to 3949. With an increase of feed concentration from 55 to 850 ppm, chloroform flux increasedlinearly but water flux remained constant, and separation factor decreased. With an increase of the feed temperaturefrom 40 to 60 oC, both flux and separation factor increased, the variation of permeation flux followed the Arrheniusrelationship, and the activation energy values were 21.65 and 9.6 KJ/mol for water and chloroform, respectively.
Li, Yang,Chen, Ling,Zhang, Yuhui,Wu, Jianmei,Lin, Yan,Fang, Zhengfeng,Che, Lianqiang,Xu, Shengyu,Wu, De Asian Australasian Association of Animal Productio 2018 Animal Bioscience Vol.31 No.6
Objective: The study was conducted to investigate the effects of replacing soybean meal (SBM) with different levels of detoxified Jatropha curcas kernel meal (DJM) in growing pig diets on growth performance, nutrients digestibility and meat edibility. Methods: A total of 144 pigs with initial body weight of $20.47{\pm}1.44kg$, were randomly allocated to 6 dietary treatments with 6 replications per treatment and 4 pigs per replication for a period of 79 days. Six diets (DJM0, DJM15, DJM30, DJM45, DJM60, and DJM75) were formulated using DJM to replace 0%, 15%, 30%, 45%, 60%, and 75% of SBM. From d 37 to 42, feces and urine were total collected from six barrows in each treatment. At day 79, thirty-six pigs were slaughtered for sampling. The feed intake and weight gain were recorded, while the intestinal morphology, digestive enzyme activities, nutrient digestibility and the content of residual phorbol esters in muscles were determined. Results: The results showed that increasing the replacement of SBM with DJM decreased the parameters including body weight, average daily gain, average daily feed intake, gain-to-feed ratio, weight and villus heights of duodenum, villus height and villus height/crypt depth of jejunum, digestive enzymes (protease, amylase, lipase, and trypsin) activities, and nutrients digestibility (nitrogen deposition, digestibility of nitrogen, energy digestibility, and total nitrogen utilization) (linear, p<0.05; quadratic, p<0.05) and there was no significant difference among DJM0, DJM15, and DJM30 in all measured indices. The highest diarrhea morbidity was observed in DJM75 (p<0.05). Phorbol esters were not detected in pig muscle tissues. Conclusion: The DJM was a good protein source for pigs, and could be used to replace SBM up to 30% (diet phorbol esters concentration at 5.5 mg/kg) in growing pig diets with no detrimental impacts on growth performance, nutrient utilization, and meat edibility.
Gong-De Yang,Ming-Yao Lin,Nian Li,Li Hao 대한전기학회 2019 Journal of Electrical Engineering & Technology Vol.14 No.1
Owing to the estimated permanent magnet (PM) flux linkage fluctuation, the stator-PM memory machine employing the continuous magnetization state (MS) manipulation may suffer from frequent MS manipulations and the accidental inverter damage in its extended speed range. In order to deal with this issue, in this paper, a novel vector control based on three MS manipulations is proposed and implemented on the existing hybrid PM axial field flux-switching memory machine. After a brief analysis of the researched machine configuration, the principle of the three MS manipulations, the remedial sliding mode speed regulator and the current distribution strategy are discussed. The simulated results show that the proposed scheme reduces the speed and electromagnetic torque overshoot and improves the dynamic performance. Meanwhile, compared with the flux-weakening control, the wide speed range can be obtained. Finally, the experiment is carried out to verify the validity of the theory.
Gong-De Yang,Xinghe Fu,Mingyao Lin,Nian Li,Hao Liu 전력전자학회 2019 JOURNAL OF POWER ELECTRONICS Vol.19 No.1
This research comparatively studies three kinds of flux regulation methods, namely, stored capacitor discharge pulse (SCDP),constant current source pulse (CCSP), and quantitative flux regulation pulse (QFRP), which are used for hybrid permanentmagnet (PM) axial field flux-switching memory machines (HPM-AFFSMMs). Through an analysis of the operation principleand the series hybrid PM flux regulation mechanism of the objective machine, the circuit topologies and flux regulation processof these flux regulation methods are addressed in detail. On the basis of a simulation, the flux regulation characteristics of theresearched machine during the magnetization and demagnetization processes are comparatively evaluated. Then, machineperformance, including back EMF, direct and quadrature axis inductances, and magnetization and demagnetizationcharacteristics, is quantitatively investigated. Results show that the QFRP enables the HPM-AFFSMM to achieve a lessharmonic component of back EMF by approximately 7.28% and 7.97% at the magnetization and demagnetization states,respectively, and a more complete magnetization process than the SCDP and CCSP.
Xiao-Lin Luo,Ya-Shao Chen,Min-Juan Wang,De-Suo Yang,Jie Yang 한국공업화학회 2015 Journal of Industrial and Engineering Chemistry Vol.32 No.-
Cu2O micro-crystals with different morphologies (including three branching structures) weresynthesized through hydrothermal method by using sodium tartrate as chelating reagent. Branchinggrowth patterns of Cu2O microcrystals have a strong dependence on the amount of sodium tartrate. These different Cu2O microcrystals were used as catalysts to promote the thermal decomposition ofammonium perchlorate (AP). The thermal decomposition of AP in the presence or absence of Cu2Omicro-crystals was investigated non-isothermally through thermogravimetry and differential scanningcalorimetry (DSC). The data obtained from DSC were applied for the calculation and comparison of thekinetic parameters of AP decomposition process through a model-free approach.
First records of two species of the genus Brachionycha H?ner (Lepidoptera: Noctuidae) in China
Qing-Yin YANG,Cheng-De LI,Hui-Lin HAN 한국곤충학회 2007 Entomological Research Vol.37 No.4
Two species of the genus Brachionycha Hbner -B. nubeculosa (Esper) and B. albicilia Sugi - are recorded for the first time from China. The adults and genital characteristics of the species are briefly redescribed with illustrations, and their distributions are given.