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Nalidixic Acid Prodrugs: Amides from amino acid ester and nalidixic acid
Taori, Ashish,Nema, Rajesh,Kohli, D.V.,Uppadhyay, R.K. The Pharmaceutical Society of Korea 1991 Archives of Pharmacal Research Vol.14 No.1
Amides from amino acid ester and nalidixic acid were synthesized. The solubility characteristics and partition coefficient of the compounds were studied. The hydrolysis of the compounds was studied in the simulated gastric fluid and simulated intestinal fluid. Some compounds showed better antibacterial activity than nalidixic acid.
A Rare Case of Male Primary Breast Lymphoma
Jawahar Rathod,Kishor Taori,Amit Disawal,Prajwaleet Gour,Suresh Dhakate,Rachna Mone,Krishna Prasad Bellam 한국유방암학회 2011 Journal of breast cancer Vol.14 No.4
Primary lymphoma of the breast is a rare occurrence because of the paucity of lymphoid tissue in the breast and is an even rarer entity in the male breast. Imaging, along with tissue diagnosis goes a long way in diagnosing breast lymphoma which has a significantly different management scheme than other breast neoplasms with respect to radio-chemotherapy rather than surgical resection. We present a case of primary male breast lymphoma which was evaluated with magnetic resonance imaging as well as other conventional imaging modalities and was treated by chemotherapy with a 7-month follow-up.
Husain, Aliabbas A.,Daginawala, Hatim F.,Warke, Shubangi R.,Kalorey, Devanand R.,Kurkure, Nitin V.,Purohit, Hemant J.,Taori, Girdhar M.,Kashyap, Rajpal S. The Korean Association of Immunobiologists 2015 Immune Network Vol.15 No.2
Evaluation and screening of vaccines against tuberculosis depends on development of proper cost effective disease models along with identification of different immune markers that can be used as surrogate endpoints of protection in preclinical and clinical studies. The objective of the present study was therefore evaluation of subcutaneous model of M.tuberculosis infection along with investigation of different immune biomarkers of tuberculosis infection in BALB/c mice. Groups of mice were infected subcutaneously with two different doses : high ($2{\times}10^6CFU$) and low doses ($2{\times}10^2CFU$) of M.tuberculosis and immune markers including humoral and cellular markers were evaluated 30 days post M.tuberculosis infections. Based on results, we found that high dose of subcutaneous infection produced chronic disease with significant (p<0.001) production of immune markers of infection like $IFN{\gamma}$, heat shock antigens (65, 71) and antibody titres against panel of M.tuberculosis antigens (ESAT-6, CFP-10, Ag85B, 45kDa, GroES, Hsp-16) all of which correlated with high bacterial burden in lungs and spleen. To conclude high dose of subcutaneous infection produces chronic TB infection in mice and can be used as convenient alternative to aerosol models in resource limited settings. Moreover assessment of immune markers namely mycobacterial antigens and antibodies can provide us valuable insights on modulation of immune response post infection. However further investigations along with optimization of study protocols are needed to justify the outcome of present study and establish such markers as surrogate endpoints of vaccine protection in preclinical and clinical studies in future.
Performance evaluation using reduced neighbor lists in cellular based multi-hop relay network
Hun-je Yeon,Eunhyun Kwon,Sung-gook Lim,Jaiyong Lee,Mi-Sun Do,Rakesh Taori 대한전자공학회 2008 ITC-CSCC :International Technical Conference on Ci Vol.2008 No.7
In this paper, we introduce neighbor list composition scheme that organizes small numbers of adjacent neighbors for cellular based multi-hop relay network so that the neighbor advertisement with small number of neighbors could increase average transmission rate of MR network. Wireless multi-hop environment based on cellular system, such as 802.16j, requires an algorithm that organizes neighbor lists dynamically due to the mobility and impermanancy of relay station. From the study, we’ve concluded that the location based neighbor lists composition could reduces the wastage of wireless resources, which improves the transmission rate of cellular based wireless multi-hop network.
Aliabbas A. Husain,Hatim F. Daginawala,Shubangi R Warke,Devanand R Kalorey,Nitin V. Kurkure,Hemant J Purohit,Girdhar M Taori,Rajpal S Kashyap 대한면역학회 2015 Immune Network Vol.15 No.2
Evaluation and screening of vaccines against tuberculosis depends on development of proper cost effective disease models along with identification of different immune markers that can be used as surrogate endpoints of protection in preclinical and clinical studies. The objective of the present study was therefore evaluation of subcutaneous model of M.tuberculosis infection along with investigation of different immune biomarkers of tuberculosis infection in BALB/c mice. Groups of mice were infected subcutaneously with two different doses : high (2×106 CFU) and low doses (2×102 CFU) of M.tuberculosis and immune markers including humoral and cellular markers were evaluated 30 days post M.tuberculosis infections. Based on results, we found that high dose of subcutaneous infection produced chronic disease with significant (p<0.001) production of immune markers of infection like IFNγ, heat shock antigens (65, 71) and antibody titres against panel of M.tuberculosis antigens (ESAT-6, CFP-10, Ag85B, 45kDa, GroES, Hsp-16) all of which correlated with high bacterial burden in lungs and spleen. To conclude high dose of subcutaneous infection produces chronic TB infection in mice and can be used as convenient alternative to aerosol models in resource limited settings. Moreover assessment of immune markers namely mycobacterial antigens and antibodies can provide us valuable insights on modulation of immune response post infection. However further investigations along with optimization of study protocols are needed to justify the outcome of present study and establish such markers as surrogate endpoints of vaccine protection in preclinical and clinical studies in future.