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Amgad I. M. Khedr,Sabrin R. M. Ibrahim,Gamal A. Mohamed,Hany E. A. Ahmed,Amany S. Ahmad,Mahmoud A. Ramadan,Atef E. Abd El-Baky,Koji Yamada,Samir A. Ross 대한약학회 2016 Archives of Pharmacal Research Vol.39 No.7
Phytochemical investigation of Ficus pandurataHance (Moraceae) fruits has led to the isolation of two newtriterpenoids, ficupanduratin A [1b-hydroxy-3b-acetoxy-11a-methoxy-urs-12-ene] (11) and ficupanduratin B [21ahydroxy-3b-acetoxy-11a-methoxy-urs-12-ene] (17), alongwith 20 known compounds: a-amyrin acetate (1), a-amyrin(2), 3b-acetoxy-20-taraxasten-22-one (3), 3b-acetoxy-11amethoxy-olean-12-ene (4), 3b-acetoxy-11a-methoxy-12-ursene (5), 11-oxo-a-amyrin acetate (6), 11-oxo-b-amyrinacetate (7), palmitic acid (8), stigmast-4,22-diene-3,6-dione(9), stigmast-4-ene-3,6-dione (10), stigmasterol (12), b-sitosterol(13), stigmast-22-ene-3,6-dione (14), stigmastane-3,6-dione (15), 3b,21b-dihydroxy-11a-methoxy-olean-12-ene (16), 3b-hydroxy-11a-methoxyurs-12-ene (18), 6-hydroxystigmast-4,22-diene-3-one (19), 6-hydroxystigmast-4-ene-3-one (20), 11a,21a-dihydroxy-3b-acetoxy-urs-12-ene(21), and b-sitosterol-3-O-b-D-glucopyranoside (22). Compound21 is reported for the first time from a natural source. The structures of the 20 compounds were elucidated on thebasis of IR, 1D (1H and 13C), 2D (1H–1H COSY, HSQC,HMBC and NOESY) NMR and MS spectroscopic data, inaddition to comparison with literature data. The isolatedcompounds were evaluated for their anti-microbial, antimalarial,anti-leishmanial, and cytotoxic activities. In addition,their radioligand displacement affinity on opioid andcannabinoid receptors was assessed. Compounds 4, 11, and15 exhibited good affinity towards the CB2 receptor, withdisplacement values of 69.7, 62.5 and 86.5 %, respectively. Furthermore, the binding mode of the active compounds inthe active site of the CB2 cannabinoid receptors was investigatedthrough molecular modelling.
Abdularahman B.O. Mohamed,Salwa Ibrahim Hindawi,Sameer Al-harthi,Qamre Alam,Mohammad Zubair Alam,Absarul Haque,Waseem Ahmad,Ghazi A Damanhouri 대한혈액학회 2016 Blood Research Vol.51 No.4
BackgroundCharacterization of the ABO blood group at the phenotype and genotype levels is clinically essential for transfusion, forensics, and population studies. This study elucidated ABO phenotypes and genotypes, and performed an evaluation of their distribution in in-dividuals from the western region of Saudi Arabia.MethodsOne-hundred and seven samples underwent standard serological techniques for ABO blood group phenotype analysis. ABO alleles and genotypes were identified using multi-plex polymerase chain reaction, and electrophoretic analysis was performed to evaluate the highly polymorphic ABO locus.ResultsA phenotype distribution of 37.4%, 30.8%, 24.3%, and 7.5% was found for blood groups O, A, B, and AB respectively in our study cohort. Genotype analysis identified 10 genotype combinations with the O01/O02 and A102/O02 genotypes being the most frequent with frequencies of 33.6% and 14.95%, respectively. Common genotypes such as A101/A101, A101/A102, A101/B101, B101/B101, and O01/O01 were not detected. Similarly, the rare genotypes, cis-AB01/O02, cis-AB01/O01, and cis-AB01/A102 were not found in our cohort. The most frequently observed allele was O02 (35.98%) followed by the A102 allele (17.76%). Furthermore, our findings are discussed in reference to ABO allele and geno-type frequencies found in other ethnic groups.ConclusionThe study has a significant implication on the management of blood bank and transfusion services in Saudi Arabian patients.
Ahmad M. Abu-Jrai,Ala’a H. Al-Muhtaseb,Jehad A. Yamin,Khalid A. Ibrahim,Omar A. Al-Khashman,Mouath A. Al-Shaweesh,Muhannad A. Hararah,Umer Rashid,Mohammad Ahmad,Gavin M. Walker 한국공업화학회 2014 Journal of Industrial and Engineering Chemistry Vol.20 No.4
The performance of a highly cross-linked polyethylene catalyst supported on alumina for low temperature selective catalytic reduction of NOx by unburned hydrocarbons (HCs) existing in an exhaust gas was examined at different engine conditions with the addition of exhaust-gas recirculation. The HXPE catalyst was shown to exhibit good NOx reduction activity at low temperatures (100–250℃) where the only reductant was the unburned HC, which was already present in the exhaust flow. The maximum NOx reduction of approximately 52% was achieved at a temperature of 150℃. HXPE demonstrated very good selectivity toward N2 in the majority of tested conditions ( 80%).
A Goodness of Fit Approach to Major Lifetesting Problems
Ahmad, Ibrahim A.,Alwasel, Ibrahim A.,Mugdadi, A.R. The Korean Reliability Society 2001 International Journal of Reliability and Applicati Vol.2 No.2
Lifetesting problems have been the subject of investigations for over three decades. Most suggested approaches are markedly different from those used in the related but wider goodness of fit problems. In the current investigation, it is demonstrated that a goodness of fit approach is possible in many lifetesting problems and that It results in simpler procedures that are asymptotically equivalent or better than standard ones. They may also have superior finite sample behavior. Several perennial classes are addressed here. The class of increasing failure rate (IFR) and the class of new better than used (NBU) are addressed first. In addition, we provide testing for a newer and practical class of new better than used in convex ordering (NBUC) due to Cao and Wang (1991). Other classes can be developed similarly and this point is illustrated with the classes of new better than used in expectation (NBUE) and harmonic new better than used in expectation (HNBUE).
Testing Whether New Is Better Than Used of Specified Age Using Moments Inequalities
Ahmad, Ibrahim A.,Al-Wasel, Ibrahim A. The Korean Reliability Society 2002 International Journal of Reliability and Applicati Vol.3 No.1
The class of “new better than used of a specified age” is a large and practical class of life distributions. Its properties, applicability, and testing was discussed by Hollander, Park and Proschan (1986). Their test, while remaining the yardstick for this class, suffers from weak efficiency and weak power, especially for specified ages below the average age. Thus, it is beneficial to have an alternative testing procedure that would work better for early ages and still work well for later ages. This is exactly the subject of the current note. The test developed here is also simpler than that of Hollander, et. al. (1986).
A robust enzymeless glucose sensor based on CuO nanoseed modified electrodes
Ahmad, Rafiq,Tripathy, Nirmalya,Hahn, Yoon-Bong,Umar, Ahmad,Ibrahim, Ahmed A.,Kim, S. H. The Royal Society of Chemistry 2015 Dalton Transactions Vol.44 No.28
<P>Herein, we demonstrate the fabrication of a robust enzymeless glucose sensor based on CuO nanoseeds (CNSs) synthesized at low-temperature. The as-fabricated sensor exhibited excellent electrocatalytic ability in a wide-linear range and was further employed for the glucose concentration determined in freshly drawn mice whole blood and serum samples.</P> <P>Graphic Abstract</P><P>CuO nanoseeds were synthesized <I>via</I> a low-temperature aqueous route, for the fabrication of a robust enzymeless glucose sensor. <IMG SRC='http://pubs.rsc.org/services/images/RSCpubs.ePlatform.Service.FreeContent.ImageService.svc/ImageService/image/GA?id=c5dt01664a'> </P>
A Note on a Recent Approach to Some Life Testing Problems
Ahmad, Ibrahim A. The Korean Reliability Society 2007 International Journal of Reliability and Applicati Vol.8 No.2
In this note, some comments concerning the testing procedures for the problems of stochastic comparison, testing IFR and testing NBU ageing properties are presented showing that the tests proposed in Belzunce, Candel and Ruiz(1998) are cumbersome to calculate and do not have as good asymptotic Pittman efficacies as simpler others already in the literature. This is done via new presentations of the measures on which Belzunce et al. base their tests.