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Pulla, R.K.,Lee, O.R.,In, J.G.,Kim, Y.J.,Senthil, K.,Yang, D.C. Academic Press 2010 Physiological and molecular plant pathology Vol.74 No.5
A full-length sequence (PgPR10-2) of the most abundant transcript from 14-year-old ginseng EST library was isolated and cloned. PgPR10-2 gene encodes 465 bp open reading frame and its deduced protein contains 155 amino acids. Genomic DNA sequence reveals it contains two exons interrupted by one intron. Expression of PgPR10-2 gene was especially abundant in roots and its transcripts showed differentially upregulated patterns against several given pathogens and abiotic stimuli. Observed enhanced ribonuclease activity and antifungal activity from tobacco transgenic lines suggest that the possible involvement of PgPR10-2 in defense-related mechanism via ribonuclease activity against biotic and abiotic stresses.
Synthesis and Evaluation of Benzimidazole Analogs as NF-κB Inhibitors
Pulla Reddy Boggu 충남대학교 약학대학 의약품개발연구소 2018 藥學論文集 Vol.33 No.-
The inhibitory in vitro activity against LPS induced NF-KB bioactivaton in RAW 264.7 cell using the SEAP assay of the substituted 2-benzylbenzimidazole analogs were investigated. Among them, (5-methoxy- 1H-benzo[이imidazol-2-yl)(4-methoxyphenyl)methanol (2b, IC50=8.4 μM) showed strong inhibition. The SAR studies 「evealed that the 5-methoxy group at phenyl ring A with additional benzylic hydroxyl group is important f。「the activity of these compounds.
Identification of novel 2-benzyl-1-indanone analogs as interleukin-5 inhibitors
Boggu, Pulla Reddy,Cho, Jungsuk,Kim, Youngsoo,Jung, Sang-Hun Elsevier 2018 European journal of medicinal chemistry Vol.152 No.-
<P><B>Abstract</B></P> <P>A novel series of 2-benzyl-1-indanone analogs were investigated as IL-5 inhibitory activity. Among the synthesized compounds, 7-(cyclohexylmethoxy)-2-(4-hydroxybenzyl)-2,3-dihydro-1<I>H</I>-inden-1-one (<B>7s</B>, 100.0% inhibition at 30 μM, IC<SUB>50</SUB> = 4.0 μM), and 7-(cyclohexylmethoxy)-2-(3-hydroxybenzyl)-2,3-dihydro-1<I>H</I>-inden-1-one (<B>7t</B>, 95.0% inhibition at 30 μM, IC<SUB>50</SUB> = 6.0 μM) showed the best inhibitory activity against IL-5. The 2-benzyl-1-indanone analogs showed moderate to strong IL-5 inhibitory activity. Especially, hydroxyl (HBD/HBA) substituent at position 3 or 4 on phenyl ring B showed potent IL-5 inhibition. Additionally, the bulky hydrophobic cyclohexylmethoxy group at position 7 of the 1-indanone ring is favorable for the inhibitory activity.</P> <P><B>Highlights</B></P> <P> <UL> <LI> Novel 2-benzyl-1-indanone scaffold has been discovered as highly active interleukin-5 inhibitor. </LI> <LI> SAR study explored the importance of hydrophobic group at position 7 and 4-hydoxybenzyl group. </LI> <LI> IC<SUB>50</SUB> values of <B>7s</B> and <B>7t</B> shows 4.0 and 6.0 μM, respectively. </LI> <LI> The conformational study indicates that the folded conformation of <B>7s</B> could be the effective conformation. </LI> </UL> </P> <P><B>Graphical abstract</B></P> <P>[DISPLAY OMISSION]</P>
Challenges and Dilemmas of Civil Society movements in India
Venkat Pulla,Neelmani Jaysawal,Sudeshna Saha 한국사회복지학회 2019 Asian Social Work and Policy Review Vol.13 No.2
Civil Society spaces provide citizens opportunities to frame their collective identities and interests through the formation of voluntary interest groups and organisations set to specific purposes. In the west, historically these interest groups have contrib-uted to the development of political thought that assisted to forge the economic interests of emerging bourgeoisie. This paper situated in the context of India begins with a thematic perspective and reviews the challenges that emerge as a result of the demands that emerge within the civil society space. The paper considered three broad range organizations for this review such as the Narmada Bachao Andolan (Save the river Narmada Campaign); National Alliance for People's Movement (NAPM); and the Self-Employed Women's Association (SEWA). The authors see civil society as a conciliating place—where individual interests appear to mingle with societal require-ments while providing adequate representation to the marginalized groups and ex-pression of concerns around economic and environmental rights.