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Pharmasol 基劑를 使用한 Indomethacin 結晶多形의 直腸吸收에 關한 硏究
이동호,김재백,Lee, D.H. 圓光大學校 藥品硏究所 1986 藥品硏究所報 Vol.1 No.1
Suppositories may be particulary important where a drug cannot be tolerated orally, where the patient cannot swallow, or where the drug may be decomposed or inactivated by the pH and enzyme present in the gastrointestinal tracts Rectal suppositories are used for the introduction of medicaments to be adsorbed into the circulatory system. In order to study on the bioavailability of Acetaminophen rectal suppository. we make two types of suppository; one is a new gelatin capsule (Rectocap) and the other is common suppository (Rectal suppository) After the rectal administration of Rectocap and Rectal suppository, we experiment the serum concentration of Acetaminophen by High Pressure Liquid Chromatography. In serum concentration, the Rectocap is higher and persisted longer than the Rectal suppository This greater serum concentration of Rectocap may be related to a variery of factors including point, the solubility chemical reactivity and the composition in the suppository bases.