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의약품 동족체 합성에 있어서 Sequential Simplex Method의 이용
한석규 부산대학교 1975 論文集 Vol.19 No.2
The utility of the sequential simplex method in designing drug analogs was examined, using 9 analog systems. The three compounds for the starting simplex were selected from Topliss operational scheme. The statistical analysis showed that the use of the method is more effective than an unsystematic choice in reaching the structure of the maximum activity at a significance level of 1%.