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( Kanika Patel ),( Dinesh Kumar Patel ) 대한간학회 2020 춘·추계 학술대회 (KASL) Vol.2020 No.1
Aims: Nature is the source of all the materials we need for the betterment of our own health in terms of food and medicine. Anthocyanins are coloured compounds responsible for various attractive colour of plant material and showed wide range of pharmacological activities. Delphinidin were present in all the bright colored fruits and vegetables which have been used in the diet as supplements for the treatment of Hepatic disorders. Methods: Present research work aim is to describe the medicinal importance and pharmacological activities of delphinidin. To know the medicinal important of delphinidin, various scientific databases have been searched and analyzed for their Health beneficial properties. Hepatoprotective activity of delphinidin has been also analyzed through various In-vivo and In-vitro experimental works in the present work. All the presented data have been analyzed through statistical method to get significant result of their Hepatoprotective activity. In-silico molecular study has been also performed for delphinidin with different ligands to search better molecular mechanism for their Hepatoprotective activity. Results: From the analysis of the presented data in this work we can reveal the importance of delphinidin in the nature. Delphinidin is an important anthocyanidins which are mainly present in the epidermal tissues of flowers and fruits. Pharmacological study revealed their importance as antioxidant, antimutagenesis, anti-inflammatory and antiangiogenic activity. The mode of mechanism of delphinidin is mainly through the vascular endothelial growth factor receptor-2 phosphorylation inhibition, platelet-derived growth factor receptor signaling, cancer cell proliferation and modulation of Met receptor phosphorylation. Delphinidin attenuated oxidative stress, increased matrix metalloproteinase- 9 and metallothionein I/II expression and restored hepatic cellular damage in the carbon tetrachloride-induced liver fibrosis with strong enhancement of hepatic regenerative power. Delphinidin showed significant scavenging activity against different free radicals. Conclusions: This work will be benificial to the scientist, manufacturer and consumers in order to explore the Hepatoprotective potential of delphinidin.