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Muthusami, Sridhar,Prabakaran, D S,Yu, Jae-Ran,Park, Woo-Yoon Springer-Verlag 2015 JOURNAL OF CANCER RESEARCH AND CLINICAL ONCOLOGY Vol.141 No.2
<P>Radiation-induced nuclear stabilization and phosphorylation of epidermal growth factor receptor (EGFR) confers radioresistance. Understanding of the factor(s) regulating the nuclear stabilization and phosphorylation of EGFR is important for the modulation of radioresistance. Present study was designed to delineate the regulation of EGFR nuclear stabilization and phosphorylation by fused toes homolog (FTS), an oncoprotein, which is responsible for the radioresistance in cervical cancer cells.</P>
Kamalakannan Reena,MANI GAJENDIRAN,Muthusamy Prabakaran,Susaimanickam Arul Antony,김교범 한국공업화학회 2017 Journal of Industrial and Engineering Chemistry Vol.51 No.-
The purpose of the study was to develop caffeine-loaded gold nanoparticles (AuNPs) using a poly(lacticacid)-polyethylene glycol-poly(lactic acid) (PLA-PEG-PLA) polymer to enhance the anti-inflammatoryactivity of caffeine. Caffeine-loaded AuNPs were conjugated to PLA-PEG-PLA copolymer matrix viap-back bond between AuNPs and the ester carbonyl group of the polyester. The p-back bonded estercarbonyl oxygen strongly interacted with the caffeine molecule and exhibited enhanced antiinflammatoryactivity. The physico-chemical characteristics of the resulting nanoconjugates wereevaluated by a series of microscopic, diffraction, and spectroscopic methods. In vitro assays indicatedincreasing membrane stabilization of red blood cells and enhanced inhibition of protein denaturation