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Momoko Nishimaru,Shoji Kudo,Hiroshi Takiyama 한국공업화학회 2016 Journal of Industrial and Engineering Chemistry Vol.36 No.-
The cocrystallization operation has the deposition risk of undesired crystals. In this study, the strategy ofcocrystal production method considering the risk reduction of undesired single component crystaldeposition was investigated. The anti-solvent cocrystallization was carried out in four-componentsystem of carbamazepine (CBZ), saccharin (SAC), methanol and water. The undesired single componentcrystals precipitated depending on the solution addition sequences. Considering the driving force foreach component, a domain without the deposition risk of the undesired crystals was determined on thephase diagram. It is important to keep the operation point in this domain for production of desiredcocrystals.