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Murat SÜKÜROGLU,Burcu ÇALISKAN ERGÜN,Serdar ?L?,M. Fethi SAHIN,Esra K?ELI,Erdem YESILADA,Erden BANOGLU 대한약학회 2005 Archives of Pharmacal Research Vol.28 No.5
A series of structurally diverse amide derivatives of [6-(3,5-dimethyl-4-chloro-pyrazole-1-yl)- 3(2H)-pyridazinone-2-yl]acetic acid were prepared and tested for their in vivo analgesic and anti-inflammatory activity by using p-benzoquinone-induced writhing test and carrageenaninduced hind paw edema model, respectively. The analgesic and anti-inflammatory activity of the compounds, 7c, 7d and 7k were found to be equipotent to aspirin (as an analgesic) and indometacin (as an anti-inflammatory drug), respectively. The other amide derivatives generally resulted in lower activity on comparision with reference compounds.