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최윤정(Yun Jung Choi),윤서영(Seo Young Yoon),최지영(Ji Young Choi),우태선(Tae Seon Woo),손건호(Kun Ho Son),이용수(Yong Soo Lee),정재훈(Jae Hoon Cheong) 대한약학회 2011 약학회지 Vol.55 No.3
The aim of this study is to evaluate the sedative effects of ethanol extract and the three major constituents of Cimicifugae Rhizoma. They decreased locomotor activity significantly, and enhanced sleeping duration induced by thiopental sodium. The ethanol extract of Cimicifugae rhizoma and 24-epi-7,8-didehydrocimigenol-3-xyloside (24-epi.) increased the Cl- influx into the intracellular area of SH-SY5Y neuroblastoma cells significantly. The present results demonstrate that the sedative effects of Cimicifugae rhizoma are mediated via the GABA-gated Cl- channel, partly by 24-epi.